June 2022
Volume 63, Issue 7
Open Access
ARVO Annual Meeting Abstract  |   June 2022
The Efficacy of Phentolamine Ophthalmic Solution and Low-Dose Pilocarpine to Improve Distance-Corrected Intermediate Visual Acuity in Patients with Presbyopia
Author Affiliations & Notes
  • Jay Stuart Pepose
    Pepose Vision Institute, Chesterfield, Missouri, United States
  • Ajay Kolli
    Ocuphire Pharma, Michigan, United States
  • Ronil Patel
    Ocuphire Pharma, Michigan, United States
  • Kavon Rahmani
    Ocuphire Pharma, Michigan, United States
  • Mina Sooch
    Ocuphire Pharma, Michigan, United States
  • Mitchell G Brigell
    Ocuphire Pharma, Michigan, United States
  • Eliot Lazar
    Ocuphire Pharma, Michigan, United States
  • Footnotes
    Commercial Relationships   Jay Pepose Acufocus, Allergan, J&J Vision, Keeler, LensGen, Mimetogen, Novartis, Ocunexis, Ocuphire Pharma, Stuart Therapeutics, Sun Pharma, Thea Pharma, Code C (Consultant/Contractor), Apellis, Ocuphire Pharma, Code I (Personal Financial Interest), Ocuphire Pharma, Code S (non-remunerative); Ajay Kolli Ocuphire Pharma, Code C (Consultant/Contractor); Ronil Patel Ocuphire Pharma, Code E (Employment); Kavon Rahmani Ocuphire Pharma, Code C (Consultant/Contractor); Mina Sooch Ocuphire Pharma, Code E (Employment); Mitchell Brigell Ocuphire Pharma, Code C (Consultant/Contractor); Eliot Lazar Ocuphire Pharma, Code C (Consultant/Contractor)
  • Footnotes
    Support  Ocuphire Pharma
Investigative Ophthalmology & Visual Science June 2022, Vol.63, 1809 – F0425. doi:
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      Jay Stuart Pepose, Ajay Kolli, Ronil Patel, Kavon Rahmani, Mina Sooch, Mitchell G Brigell, Eliot Lazar; The Efficacy of Phentolamine Ophthalmic Solution and Low-Dose Pilocarpine to Improve Distance-Corrected Intermediate Visual Acuity in Patients with Presbyopia. Invest. Ophthalmol. Vis. Sci. 2022;63(7):1809 – F0425.

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      © ARVO (1962-2015); The Authors (2016-present)

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Abstract

Purpose :
The objective of this study is to evaluate the efficacy of a combination of 0.75% phentolamine ophthalmic solution (POS) and 0.4% low-dose pilocarpine (LDP) to improve distance-corrected intermediate visual acuity (DCIVA) in patients with presbyopia.

Methods : The VEGA-1 study is a Phase 2, multi-center, randomized, placebo-controlled, double-masked clinical trial. Subjects with distance-corrected near visual acuity (DCNVA) of 20/50 or worse were randomized to receive either 0.75% POS or placebo vehicle in the evening, followed with and without a morning dose of 0.4% LDP. DCIVA was assessed at multiple time points after a single combination treatment. Logistic regression models comparing POS+LDP to each treatment, with treatment and light/dark irides as factors and baseline DCIVA as a covariate was used to compare the proportion of patients with 5-letter and 10-letter improvements in DCIVA. Mean improvements in DCIVA were also assessed.

Results : Of the 150 participants included in this clinical trial (mean age 53.1 years, 72% female, 89% White), 43 were randomized to placebo alone, 30 to POS alone, 43 to POS+LDP, and 30 to LDP alone. Subjects treated with POS+LDP had a mean (SD) 9.6 (5.7) letter improvement in DCIVA from baseline at 1 hour vs 4.5 (6.7) letters with placebo (p<0.0001). This improvement was seen in those with both irides: light 10.4 (5.7) letters; dark 8.4 (5.6) letters. At 6 hours, POS+LDP conferred a 7.1 (6.0) letter improvement from baseline, significantly more than placebo (4.0 [6.3], p<0.0001). LDP+POS yielded a greater proportion of patients with a ≥ 10-letter improvement in DCIVA than placebo at 1 hour (49% vs 27%, p=0.027). A greater proportion of patients treated with POS+LDP had ≥ 5 letter improvement in DCIVA at 1 hour compared to placebo (86% vs 58%, OR: 5.2, p=0.004) and at 6 hours (72% vs 49%, OR: 3.0, p=0.027).

Conclusions : In this Phase 2 clinical trial, 0.75% POS and 0.4% LDP significantly improved DCIVA in subjects with presbyopia at 1 hour, with durable results through 6 hours. Phase 3 studies are planned to advance POS+LDP for a potential treatment for presbyopia.

This abstract was presented at the 2022 ARVO Annual Meeting, held in Denver, CO, May 1-4, 2022, and virtually.

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