June 2023
Volume 64, Issue 8
Open Access
ARVO Annual Meeting Abstract  |   June 2023
CB13 is a mixed CB1/CB2 cannabinoid receptor agonist that protects zebrafish photoreceptors from light-induced retinal degeneration.
Author Affiliations & Notes
  • Renata Proano
    Neural and Behavioral Sciences, Penn State Health Milton S Hershey Medical Center, Hershey, Pennsylvania, United States
  • Alexandria Ostman
    Neural and Behavioral Sciences, Penn State Health Milton S Hershey Medical Center, Hershey, Pennsylvania, United States
  • Salvatore L Stella
    Neural and Behavioral Sciences, Penn State Health Milton S Hershey Medical Center, Hershey, Pennsylvania, United States
  • Footnotes
    Commercial Relationships   Renata Proano None; Alexandria Ostman None; Salvatore Stella None
  • Footnotes
    Support  None
Investigative Ophthalmology & Visual Science June 2023, Vol.64, 5226. doi:
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      Renata Proano, Alexandria Ostman, Salvatore L Stella; CB13 is a mixed CB1/CB2 cannabinoid receptor agonist that protects zebrafish photoreceptors from light-induced retinal degeneration.. Invest. Ophthalmol. Vis. Sci. 2023;64(8):5226.

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      © ARVO (1962-2015); The Authors (2016-present)

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Abstract

Purpose : Retinal diseases that damage photoreceptors, particularly those that affect cones such as the “dry” form of age-related macular degeneration (AMD), have dire consequences for vision. Models of light-induced retinal degeneration (LIRD) recapitulate some of the hallmarks of oxidative damage observed in “dry” AMD. One strategy for treatment of AMD, is to employ a “druggable” therapy targeted to neuroprotective mechanisms in photoreceptors. Cannabinoids have been shown to prevent oxidative stress-driven damage in central neurons, thus preventing neurodegeneration. The purpose of this study was to test whether targeting cannabinoid receptors could prevent light damage to photoreceptors in zebrafish retina.

Methods : Adult Tg(nrd:GFP) zebrafish (used to GFP label rod photoreceptors) were dark-adapted for 24 hrs, followed by intravitreal injections of a mixed cannabinoid receptor agonist, 1 µM CB13 (CB1/CB2). Controls were injected with saline in both eyes. All zebrafish were exposed to high-intensity light (≥ 28,000 lux) and collected at 0 and 96 hours post dark-adaptation. Immunohistochemical analysis was performed with cell specific markers, and cell death assays on zebrafish retinas in order to assess the impact of CB13 on light-induced photoreceptor damage of rods and cones.

Results : Photoreceptors treated with 96 hours of light exposure exhibited severe truncation or loss of the outer segments and swelling. Additionally, there was an increase in cell death and a significant decrease in rod and cone photoreceptors. Treatment of retinas with 1 µM CB-13 prior to light lesioning prevented cell damage, and reduced truncation of the outer segments, lacked swelling, and had morphology similar to retinas collected prior to light exposure.

Conclusions : These findings demonstrate that cannabinoids have the capacity to prevent oxidative stress-driven light damage following intense light exposure. Thus, cannabinoids could serve as a potential novel therapeutic target for the treatment of the dry form of AMD.

This abstract was presented at the 2023 ARVO Annual Meeting, held in New Orleans, LA, April 23-27, 2023.

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