June 2023
Volume 64, Issue 8
Open Access
ARVO Annual Meeting Abstract  |   June 2023
Phentolamine Ophthalmic Solution Rapidly Reverses Pharmacologically Induced Mydriasis in Two Pivotal Phase 3 MIRA Trial
Author Affiliations & Notes
  • Mina Sooch
    Ocuphire Pharma Inc, Farmington Hills, Michigan, United States
  • Jay Stuart Pepose
    Ocuphire Pharma Inc, Farmington Hills, Michigan, United States
  • Louis Haddad
    Ocuphire Pharma Inc, Farmington Hills, Michigan, United States
  • Amar Khatri
    Ocuphire Pharma Inc, Farmington Hills, Michigan, United States
  • Audrey Lazar
    Ocuphire Pharma Inc, Farmington Hills, Michigan, United States
  • Drey Coleman
    Ocuphire Pharma Inc, Farmington Hills, Michigan, United States
  • Mitchell G Brigell
    Ocuphire Pharma Inc, Farmington Hills, Michigan, United States
  • Footnotes
    Commercial Relationships   Mina Sooch Ocuphire Pharma, Code E (Employment), Ocuphire Pharma, Code I (Personal Financial Interest), Ocuphire Pharma, Code O (Owner), Ocuphire Pharma, Code P (Patent), Ocuphire Pharma, Code S (non-remunerative); Jay Pepose Ocuphire Pharma, Code C (Consultant/Contractor), Ocuphire Pharma, Code I (Personal Financial Interest), Ocuphire Pharma, Code S (non-remunerative); Louis Haddad Ocuphire Pharma, Code C (Consultant/Contractor); Amar Khatri Ocuphire Pharma, Code E (Employment); Audrey Lazar Ocuphire Pharma, Code C (Consultant/Contractor); Drey Coleman Ocuphire Pharma, Code E (Employment); Mitchell Brigell Ocuphire Pharma, Code C (Consultant/Contractor)
  • Footnotes
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Investigative Ophthalmology & Visual Science June 2023, Vol.64, 3099. doi:
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      Mina Sooch, Jay Stuart Pepose, Louis Haddad, Amar Khatri, Audrey Lazar, Drey Coleman, Mitchell G Brigell; Phentolamine Ophthalmic Solution Rapidly Reverses Pharmacologically Induced Mydriasis in Two Pivotal Phase 3 MIRA Trial. Invest. Ophthalmol. Vis. Sci. 2023;64(8):3099.

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      © ARVO (1962-2015); The Authors (2016-present)

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Abstract

Purpose : Pharmacologically induced mydriasis, a key aspect of comprehensive eye exams and procedures, can lead to photophobia, discomfort, and impairment of vision. The MIRA-2 and MIRA-3 trials assessed time savings of reversing pharmacologically induced mydriasis with 0.75% phentolamine ophthalmic solution (POS).

Methods : MIRA-2 and MIRA-3 were multi-center, randomized, placebo-controlled, double-masked clinical trials in healthy subjects (approximately n=553; age ≥12 years). Stratified by iris color, subjects were randomized to mydriatic agent 3:1:1 (2.5% phenylephrine, 1% tropicamide, or Paremyd, respectively) and POS or placebo treatment 1:1 in MIRA-2 and 2:1 in MIRA-3. The primary efficacy endpoint was the percent of subjects returning to ≤ 0.2 mm from baseline photopic pupil diameter (PD) at 90 minutes (min). A series of endpoints were evaluated in a prespecified hierarchical analysis for the integrated dataset, including time to return to baseline PD.

Results : Across MIRA-2 and MIRA-3, 338 subjects received POS (mean age 33 years, 60% female) and 215 subjects received placebo (mean age 33 years, 62% female). In addition, time to reversal of mydriasis for both study and fellow eyes overall, for each mydriatic agent, and for light and dark irides were endpoints that met statistical significance in the hierarchy. Overall, eyes treated with POS showed a significantly faster mean time to return to ≤ 0.2 mm from baseline PD compared with placebo, for study eyes and fellow eyes (2.2 vs 6.1 hr, 2.6 vs 6.3 hr, respectively; p<0.0001). Results for subjects receiving phenylephrine, tropicamide, or Paremyd were similar (1.3 vs 5.2 hr, 3.9 vs 7.6 hr, 3.0 vs 7.2 hr respectively; p<0.0001) as well as subjects with light or dark irides (1.9 vs 6.7 hr, 2.4 vs 5.5 hr respectively; p<0.0001).

Conclusions : MIRA-2 and MIRA-3 represent two well-controlled and confirmatory Phase 3 clinical trials where the primary and secondary endpoints met clinical and statistical significance. With POS, a time savings of approximately 4 hours was seen regardless of dilating agent or iris color. Based on its efficacy and favorable safety and tolerability profile, an NDA for POS has been submitted for consideration of regulatory approval for the treatment of pharmacologically-induced mydriasis

This abstract was presented at the 2023 ARVO Annual Meeting, held in New Orleans, LA, April 23-27, 2023.

 

MIRA-2 and MIRA-3 Phase 3 Trial for POS in Reversal of Mydriasis Indication

MIRA-2 and MIRA-3 Phase 3 Trial for POS in Reversal of Mydriasis Indication

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